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Pd-Catalyzed C–H aziridination of 3,3,5,5-tetrasubstituted piperazin-2-ones

A palladium mediated C–H aziridination reaction of 3,3,5,5-substituted-piperazin-2-ones has been developed using phenyliodonium diacetate (PIDA) and succinic acid to give synthetically useful bicyclic aziridines, in moderate to good yields. Succinic acid was found to be key for selectively promoting C–N bond format

Authors:   Thomas A. Alanine; Stephen Stokes; Craig A. Roberts; James. S. Scott
Journal:   Organic & Biomolecular Chemistry
DOI:   10.1039/C7OB02486J
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